Affinity DataIC50: 51.1nMAssay Description:Inhibition of human CDK18/cyclin-Y using RB protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 66.3nMAssay Description:Inhibition of human CDK18/cyclin-Y using RB protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Blocking activity against Beta-1 adrenergic receptor in spontaneously beating guinea pig atrial preparationsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Displacement of specifically bound [3H]naloxone from rat brain homogenate, in the absence of NaClMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Effective concentration required for inhibitory activity towards human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >8.00E+3nMAssay Description:Inhibition of CDK18 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human cyclinY/CDK18 T166M mutant using YRRAAVPPSPSLS as substrate measured after 40 mins in presence of [gamma3...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 54nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 44nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 1.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 2.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 270nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 1.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 510nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 270nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 270nMAssay Description:Binding constant for full-length PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for full-length PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to PCTK3More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 20nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 4.60E+3nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 8.40E+3nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 18 [3-474](Homo sapiens (Human))
Ambit Biosciences
Curated by PubChem BioAssay
Ambit Biosciences
Curated by PubChem BioAssay
Affinity DataKd: 3.20E+3nMAssay Description:Binding constant for PCTK3 kinase domainMore data for this Ligand-Target Pair